1. Signaling Pathways
  2. Antibody-drug Conjugate/ADC Related
  3. Antibody-Oligonucleotide Conjugates (AOCs)

Antibody-Oligonucleotide Conjugates (AOCs) (抗体寡核苷酸偶联物)

Antibody-Oligonucleotide Conjugate (AOC) consists of three parts: antibody, linker and oligonucleotide. AOC combines the tissue-specific targeting of antibody drugs with the target-specific capabilities of small nucleic acids, addressing the limitation of current small nucleic acid drugs that mainly target the liver through LNP and GalNAc delivery systems.

Antibody-Oligonucleotide Conjugates (AOCs) 相关产品 (3):

Cat. No. Product Name Effect Purity Chemical Structure
  • HY-177452
    Zeleciment basivarsen
    Zeleciment basivarsen (DYNE-101) 是一种抗体寡核苷酸偶联物 (AOC),由一种与肌肉细胞转铁蛋白受体1 (TfR1) 结合的 Fab 抗体 Zeleciment (HY-P990780) 与一种反义寡核苷酸 Basivarsen (HY-177453) 组成。Zeleciment basivarsen 靶向突变型 I 型肌营养不良蛋白激酶 (DMPK) 的 RNA 进行 RHase H 介导的降解,用于肌营养不良症 1 型 (DM1) 的研究。
    Zeleciment basivarsen
  • HY-177453
    Basivarsen
    Basivarsen (DYNE-101 oligomer) 由反义寡核苷酸和连接子 (HY-177454) 组成,靶向突变型 I 型肌营养不良蛋白激酶 (DMPK) 的 RNA 进行 RHase H 介导的降解,用于肌营养不良症 1 型 (DM1) 的研究。
    Basivarsen
  • HY-P990780
    Zeleciment 98.85%
    Zeleciment 是一种抗 TFRC 的 IgG1κ 单克隆抗体。
    Zeleciment